Home Tools
Log in
Cart

Search Result

Search Results for " nk1 antagonist 1 "

20

Compounds

Cat No. Product Name Synonyms Targets
T12233 NK-1 Antagonist 1 Rolapitant intermediate Others
NK-1 Antagonist 1 is a NK-1 receptor antagonist.
T6905 Netupitant Ro 67-31898/000,CID 6451149 Neurokinin receptor
Netupitant (CID 6451149) is a specific neurokinin 1 (NK1) receptor antagonist (Ki: 0.95 nM).
T13306L Vapreotide acetate RC-160 acetate,BMY-41606 acetate Neurokinin receptor
Vapreotide acetate (BMY-41606 acetate) is an antagonist of the neurokinin-1 (NK1) receptor (IC50: 330 nM).
T68068 Ezlopitant CJ 11974,CJ-11974,CJ11974 Neurokinin receptor
Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.
T3716 Rolapitant SCH619734 Neurokinin receptor
Rolapitant (SCH619734) Hydrochloride is the hydrochloride salt form of rolapitant, an orally bioavailable, centrally-acting, selective, neurokinin 1 receptor (NK1-receptor) antagonist with potential antiemetic activity. ...
T3724 Rolapitant hydrochloride Rolapitant HCl Neurokinin receptor
Rolapitant (SCH619734) hydrochloride is a potent, selective, long-acting and orally active neurokinin 1 (NK1) receptor antagonist with a K i of 0.66 nM. Rolapitant hydrochloride (Rolapitant HCl) does not interact with CY...
T28917 TAK-637 TAK 637
TAK-637 is a tachykinin 1 (NK1) receptor antagonist.
T9471 Imnopitant
Imnopitant is an antagonist of the NK1 receptor [1].
T13306 Vapreotide BMY 41606,RC160 Others
Vapreotide is an antagonist of the neurokinin-1 (NK1) receptor (IC50: 330 nM).
T10688 Casopitant mesylate GW679769B P450 , Neurokinin receptor
Casopitant mesylate (GW679769B) is a selective, brain permeable, and orally active antagonist of neurokinin 1 (NK1) receptor. It is a second in the class of antiemetics.
T73705 Imnopitant dihydrochloride
Imnopitant dihydrochloride is a neurokinin NK1 receptor antagonist [1] .
T78104 Fosnetupitant chloride monohydrochloride Pronetupitant chloride monohydrochloride Neurokinin receptor
Fosnetupitant chloride monohydrochloride (Pro-netupitant chloride monohydrochloride) is a selective NK1 antagonist exhibiting high affinity for the human NK1 receptor with a pK i value of 9.5, and a lower affinity for th...
T38033 Benzomalvin B
Benzomalvin B is a fungal metabolite originally isolated from Penicillium. It acts as an antagonist of neurokinin-1 (NK1) receptors, inhibiting binding of substance P by 24% in vitro when used at a concentration of 100 μ...
T66676 SCH619734 SCH-619734
Rolapitant Hydrochloride is the hydrochloride salt form of rolapitant, an orally bioavailable, centrally-acting, selective, neurokinin 1 receptor (NK1-receptor) antagonist with potential antiemetic activity.
T71833 Acetylaszonalenin
Acetylaszonalenin is a fungal metabolite that has been found in A. flavipes.1 It acts as an antagonist of neurokinin-1 (NK1) receptors, inhibiting binding of substance P with a Ki value of 170 μM.
T71935 WIN 66306
WIN 66306 is a cyclic heptapeptide antagonist of neurokinin-1 (NK1) and NK2 receptors originally isolated from A. flavipes. It binds to NK1 and NK2 receptors and inhibits contractions induced by substance P in isolated g...
T80031 [D-Pro2] Spantide I TFA Neurokinin receptor
[D-Pro2] Spantide I TFA is an analog of Spantide I, a selective antagonist of the NK1 receptor [1].
T70456 Nolpitantium Free Base
Nolpitantium Free Base is a highly selective nonpeptide antagonist of neurokinin-1 (NK1) receptor. Nolpitantium potently, selectively and competitively inhibited substance P binding to NK1 receptors from various animal s...
T68371 Rolapitant hydrochloride hydrate
Rolapitant, also known as SCH-619734, is an orally bioavailable, centrally-acting, selective, neurokinin 1 receptor (NK1-receptor) antagonist with potential antiemetic activity. Upon oral administration, rolapitant compe...
T75837 Spantide I TFA
Spantide I TFA, a selective NK1 receptor antagonist and a substance P analog, exhibits K(i) values of 230 nM for NK1 and 8150 nM for NK2 receptors, respectively. It offers a method to decrease type 1 while increasing typ...
1 2
TargetMol